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(11)    Patent No :    AP 2322   
(21)    Application No :    AP/P/2008/004308   
(22)    Filing Date :    26.07.2006   
(24)    Date of Grant &    18.11.2011   
(45)    Publication :

(30)  Priority Data       
(33) Country    (31) Number    (32) Date
EP    05106962.3    28.07.2005

(84)    Designated State

BW    GM    GH    KE    LS    MW  MZ   NA   SL
SD    SZ    T Z    UG    ZM    ZW

(73) Applicant(s)


B-2340 Beerse,

(72) Inventors

GUILLEMONT Jérôme Emile Georges, France

LANÇ OIS David Francis Alain, France

PASQUIER Elisabeth Thérèse Jeanne, France

et al

(74) Representative


(51)  International  Classification   A61K 31/47 (2006.01)    A61P 31/00 (2006.01)
C07D 215/12 (2006.01)   

(54)    Title

Antibacterial quinoline derivatives

(57)    Abstract

The present invention relates to novel substituted quinoline derivatives according to the general Formula (Ia) or Formula (Ib): the pharmaceutically acceptable acid or base addition salts thereof, the quaternary amines thereof, the stereochemically isomeric forms thereof, the tautomeric forms thereof and

the N-oxide forms thereof. The claimed compounds are useful for the treatment of a bacterial disease including a mycobacterial disease, particularly those diseases caused by pathogenic mycobacteria such as Mycobacterium tuberculosis, M. bovis, M. avium and M. marinum. Also claimed is a composition comprising a pharmaceutically acceptable carrier and, as active ingredient, a therapeutically effective amount of the claimed compounds, the use of the claimed compounds or compositions for the manufacture of a medicament for the treatment of bacterial diseases and a process for

(56)  Documents Cited :    WO 2004/011436


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