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(11)    Patent No :    AP 2048   
(21)    Application No :    AP/P/2005/003353   
(22)    Filing Date :    05.01.2004   
(24)    Date of Grant &    24.09.2009   
           
(45)    Publication :

(30)  Priority Data       
(33) Country    (31) Number    (32) Date
US    60/439,396    09.01.2003
(4)    Designated State

GM    GH    KE   LS   MW  MZ   SL   SD   SZ
T Z    UG    ZW

(73) Applicant(s)

PFIZER INC., 235 East 42nd Street, New York, New York 10017
United States of America

(72) Inventors

NINKOVIC Sacha, United States of America BENNETT Michael John, United States of America RUI Eugene Yuanjin, United States of America

et al

(74) Representative

GALLOWAY & COMPANY
 

(51)  International  Classification   A61K 31/55 (2006.01)    A61P 35/00 (2006.01)
C07D 487/06 (2006.01)   


(54)    Title

Diazepinoindole derivatives as kinase inhibitors

(57)    Abstract

Protein kinase, such as CHK-1, inhibiting tricyclic compounds of the following formula (wherein R2, R3 and R4 are as defined in the specification) pharmaceutical compositions containing effective amounts of said compounds or their salts are useful as a single agent or in combination with an anti-neoplastic agent or therapeutic radiation having an anti-neoplastic effect for treating diseases or conditions, such as cancers.

(56)    Documents Cited :    WO 02/44183 A   WO 00/42040 A

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